跳到正文
AACR 2026 现场信号· @ · X·· 2026-04-22评分60

FHD-909

解读

工具与平台层 — 分子胶、空间组学、AI

FHD-909 / MRT-55811 / MR-2088 · 表观 / ULK 等工具分子在会场出现

正文 · 机器翻译

在2026年 @AACR 年会上,我们公布了选择性 SMARCA2 抑制剂 FHD-909 以及选择性 CBP、EP300 和 ARID1B 降解剂项目的全新临床前数据。查看研究发现:https://t.co/eyKPNmKe2C

#AACR26 https://t.co/hX3PN7xifm

热度 1 · 1 赞 · 0 回复 · 0 转发

会议摘要
3500按 代号 EP300 对上
Synergistic targeting of EP300/CBP and EYA co-activators collapses the rhabdomyosarcoma core regulatory circuit

Annika Gustafson, Stephanie Nance, Berkley Gryder, Noha A. Shendy, Lars Wick, Grace McKay-Corkum, K. Elaine Ritter, Stephen Connor Purdy, Arthur R. Wolin, Sheera R. Rosenbaum, Sabateeshan Mathavarajah, Nickerson A. Demelfi, Yueyang Wang, Yang Zhang, Mark W. W. Zimmerman, Anoop M. Kavirayani, John Hardin, Alexander LaVeck, Xiang Wang, Neekesh V. Dharia, Andrew Hong, Guillaume Kugener, Jesse S. Boehm, Jennifer Roth, Javed Khan, Francisca Vasquez, Kristin B. Artinger, Rui Zhao, David M. Langenau, Jun Qi, Kimberly Stegmaier, Heide L. Ford, Adam D. Durbin, Brian J. Abraham

读摘要原文 →
4024按 代号 EP300 对上
Dysregulated AKT signaling reprograms osteosarcoma to drive selective reliance on EP300

Ian Delahunty, Stephanie Nance, Yang Zhang, Francois Lamoureux, Qi Liu, W. Charlie Wright, K. Elaine Ritter, Noha A. Shendy, Benedicte Brounais, Sandra Kietlinska, Barbara De Kegel, Matthew G. Rees, Mustafa Kocak, Ashish B. George, Anoop M. Kavirayani, Paris P. Prinsen, Yousef Khashana, Melissa M. Ronan, Jennifer Roth, Alejandro Sweet-Cordero, Xiaotu Ma, Lillian M. Guenther, Paul Geeleher, Benjamin Ory, Jun Qi, Brian Abraham, Adam D. Durbin

读摘要原文 →

来源:AACR 2026 现场信号 · x.com

CBACBA Frontier Insights (CFI)美国华人生物医药科技协会(CBA)www.cba-usa.org