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Yale Cancer Center· @YaleCancer · X·· 2026-04-20Score60

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KRAS / RAS targeting: from platform to Phase 3

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Newly presented #AACR26 miPEP133 emerges as a potential tumor suppressor in #ovariancancer. Restoring its expression slowed tumor cell growth and increased sensitivity to chemotherapy and MEK inhibitors.
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Conference abstracts
CT129matched by 摘要号 CT129
Preliminary results from a Phase 1a/b dose-escalation and expansion trial of the pan-RAF-MEK molecular glue NST-628 in patients (pts) with advanced or refractory RAF, KRAS, and NRAS-mutant solid tumors

Ahmad A. Tarhini, Monica Chen, Jia Liu, Varun Monga, Victoria Atkinson, Sarina A. Piha-Paul, Bartosz Chmielowski, Benjamin Herzberg, Charlotte Lemech, Prachi Bhave, Ganessan Kichenadasse, Gerald Falchook, Janice Mehnert, Andrae Vandross, Mohamad Salkeni, Meredith McKean, David Wages, Ann Marie Kennedy, Meagan B. Ryan, John Clark, Abdulaziz Nanah, Michael J. Fossler, Philip Komarnitsky, Igor Puzanov

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Source: Yale Cancer Center · x.com

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